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Assay Detail

CHEMBL749394

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of cloned human NK1 (Neurokinin 1) receptor, stably expressed in chinese hamster ovary (CHO) cells was determined
18
Total Activities
18
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Cell Type CHO
Confidence 8 — Homologous single protein target
Curated By Expert

Target

Substance-P receptor (CHEMBL249)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

L-tryptophan urea amides as NK1/NK2 dual antagonists.
Qi H, Shah SK, Cascieri MA, Sadowski SJ, MaCcoss M.
Bioorg Med Chem Lett (1998) 8 : 2259 -2262
PubMed 9873524 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 18 7.29 9.24

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL72234 1 9.24
CHEMBL306400 1 9.00
CHEMBL22870 L-732138 1 8.80
CHEMBL74237 1 8.00
CHEMBL306065 1 7.85
CHEMBL73097 1 7.64
CHEMBL73618 1 7.25
CHEMBL305509 1 7.17
CHEMBL73839 1 7.11
CHEMBL23851 1 6.99
CHEMBL2114103 1 6.79
CHEMBL303868 1 6.64
CHEMBL73896 1 6.62
CHEMBL74176 1 6.48
CHEMBL305609 1 6.32
CHEMBL308148 SAREDUTANT 3.0 1 6.10
CHEMBL70461 1 5.96
CHEMBL305608 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL72234 IC50 = 0.58 nM 9.24
CHEMBL306400 IC50 = 1.0 nM 9.00
CHEMBL22870 L-732138 IC50 = 1.6 nM 8.80
CHEMBL74237 IC50 = 10.0 nM 8.00
CHEMBL306065 IC50 = 14.0 nM 7.85
CHEMBL73097 IC50 = 23.0 nM 7.64
CHEMBL73618 IC50 = 56.0 nM 7.25
CHEMBL305509 IC50 = 68.0 nM 7.17
CHEMBL73839 IC50 = 77.0 nM 7.11
CHEMBL23851 IC50 = 103.0 nM 6.99
CHEMBL2114103 IC50 = 164.0 nM 6.79
CHEMBL303868 IC50 = 227.0 nM 6.64
CHEMBL73896 IC50 = 242.0 nM 6.62
CHEMBL74176 IC50 = 332.0 nM 6.48
CHEMBL305609 IC50 = 480.0 nM 6.32
CHEMBL308148 SAREDUTANT IC50 = 800.0 nM 6.10
CHEMBL70461 IC50 = 1100.0 nM 5.96
CHEMBL305608 IC50 > 1100.0 nM -