Assay Detail
Functional
CHEMBL749485
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Evaluated for its antagonistic activity against the NT-stimulated cyclic [3H]GMP formation in murine N1E-115 neuroblastoma cells
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Cell Type | N1E-115 |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
UK-73,093: A non-peptide neurotensin receptor antagonist
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 5.36 | 5.36 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL38243 | — | — | 1 | 5.36 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL38243 | — | Ki | = | 4400.0 | nM | 5.36 |