Assay Detail
Functional
CHEMBL750982
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antagonist activity against recombinant human P2X purinoceptor 4 (P2X4)
8
Total Activities
8
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
Purine and pyrimidine (P2) receptors as drug targets.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 8 | 5.46 | 6.31 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL339386 | — | — | 1 | 6.31 |
| CHEMBL14249 | ADENOSINE TRIPHOSPHATE | 2.0 | 1 | 6.30 |
| CHEMBL336208 | — | — | 1 | 6.00 |
| CHEMBL339385 | DIADENOSINE TETRAPHOSPHATE | — | 1 | 6.00 |
| CHEMBL69234 | — | — | 1 | 5.00 |
| CHEMBL335206 | — | — | 1 | 4.60 |
| CHEMBL28324 | — | — | 1 | 4.00 |
| CHEMBL223344 | RB 2 | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL339386 | — | EC50 | = | 490.0 | nM | 6.31 |
| CHEMBL14249 | ADENOSINE TRIPHOSPHATE | EC50 | = | 500.0 | nM | 6.30 |
| CHEMBL336208 | — | EC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL339385 | DIADENOSINE TETRAPHOSPHATE | EC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL69234 | — | EC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL335206 | — | EC50 | = | 25000.0 | nM | 4.60 |
| CHEMBL28324 | — | EC50 | = | 100000.0 | nM | 4.00 |
| CHEMBL223344 | RB 2 | EC50 | = | 128000.0 | nM | - |