Assay Detail

CHEMBL751771

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Binding

Dissociative constant at P2Y purinoceptor 1 (P2Y1) from guinea pig taenia coli

ChEMBL ↗

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Target

P2Y purinoceptor 1 (CHEMBL4315) ↗

Open DB target context

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P2Y purinoceptor 1 (CHEMBL4315) is the working anchor for this assay review. Loading the live Open DB target snapshot…

Primary target P2Y purinoceptor 1

CHEMBL4315

Anchored from Assay target.

Protein identity P2Y purinoceptor 1

Disease frame Disease evidence pending

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Review focus Open DB context pending

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Total Activities

Compounds Tested

Activity Types

Assay Parameters

Assay Information

Assay Type	Binding
Organism	Cavia porcellus
Confidence	8 — Homologous single protein target
Curated By	Autocuration

Target

P2Y purinoceptor 1 (CHEMBL4315) ↗

Type	SINGLE PROTEIN
Organism	Homo sapiens

Publication

Purine and pyrimidine (P2) receptors as drug targets.

Jacobson KA, Jarvis MF, Williams M.
J Med Chem (2002) 45 : 4057 -4093
PubMed 12213051 · DOI

Activity Statistics

Type	Count	Avg pChEMBL	Best pChEMBL
Kd	1	5.85	5.85

Compounds Tested

Compound	Name	Phase	Activities	Best pChEMBL
CHEMBL133576	ACID BLUE 129	—	1	5.85

Activity Data

Compound	Name	Type	Rel.	Value	Units	pChEMBL
CHEMBL133576	ACID BLUE 129	Kd	=	1400.0	nM	5.85