Assay Detail
Functional
CHEMBL751808
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The compound was evaluated for antagonist activity against recombinant human P2X purinoceptor 3 (P2X3 )
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Purine and pyrimidine (P2) receptors as drug targets.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.81 | 7.08 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL69727 | ISOPPADS | — | 1 | 7.08 |
| CHEMBL216504 | — | — | 1 | 4.54 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL69727 | ISOPPADS | IC50 | = | 84.0 | nM | 7.08 |
| CHEMBL216504 | — | IC50 | = | 28500.0 | nM | 4.54 |