Assay Detail
Binding
CHEMBL753770
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Binding affinity towards Opioid receptor mu 1 using [3H]DAMGO expressed as Kd
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
N-Methyl and N-cyclopropylmethyl-14,14-[dithiobis[(2-oxo-2,1-ethanediyl)imino]]bis(7,8-dihydro-5-methyl-morphinone) MET-TAMO and N-CPM-MET-TAMO: Synthesis and opioid binding properties
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 1 | 9.40 | 9.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2304424 | — | — | 1 | 9.40 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2304424 | — | Kd | = | 0.4 | nM | 9.40 |