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Assay Detail

CHEMBL754604

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity (in vitro) against Opioid receptor delta 1 using radio-ligand binding assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Delta-type opioid receptor (CHEMBL4103)
Type SINGLE PROTEIN
Organism Sus scrofa

Publication

Semisynthetic preparation of amentoflavone: A negative modulator at GABA(A) receptors.
Hanrahan JR, Chebib M, Davucheron NL, Hall BJ, Johnston GA.
Bioorg Med Chem Lett (2003) 13 : 2281 -2284
PubMed 12824018 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 7.44 7.44

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL63354 AMENTOFLAVONE 1 7.44

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL63354 AMENTOFLAVONE Ki = 36.5 nM 7.44