Assay Detail
Binding
CHEMBL754642
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Compound was tested for the inhibition of inducible murine macrophage nitric oxide(NO) synthase, activity expressed as inhibitory constant
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
NG-allyl- and NG-cyclopropyl-L-arginine: two novel inhibitors of macrophage nitric oxide synthase.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 5.43 | 5.47 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL106425 | 5-N-ALLYL-ARGININE | — | 1 | 5.47 |
| CHEMBL256147 | TILARGININE | 3.0 | 1 | 5.38 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL106425 | 5-N-ALLYL-ARGININE | Ki | = | 3400.0 | nM | 5.47 |
| CHEMBL256147 | TILARGININE | Ki | = | 4200.0 | nM | 5.38 |