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Assay Detail

CHEMBL754784

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Compound was tested in vitro for its binding affinity against Neurotensin Receptor after peripheral administration
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Neurotensin receptor type 1 (CHEMBL3570)
Type SINGLE PROTEIN
Organism Mus musculus

Publication

Reduced amide bond neurotensin 813 mimetics with potent in vivo activity
Wustrow D, Davis M, Akunne H, Corbin A, Wiley J, Wise L, Heffner T
Bioorg Med Chem Lett (1995) 5 : 997 -1002
· DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 10.19 10.19

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL266571 1 10.19

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL266571 Ki = 0.064 nM 10.19