Assay Detail
Binding
CHEMBL756174
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Binding affinity towards Opioid receptor delta 1 was evaluated
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Enkephalin glycopeptide analogues produce analgesia with reduced dependence liability.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 8.55 | 8.62 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1790710 | — | — | 1 | 8.62 |
| CHEMBL1790709 | — | — | 1 | 8.47 |
| CHEMBL70 | MORPHINE | 4.0 | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1790710 | — | IC50 | = | 2.4 | nM | 8.62 |
| CHEMBL1790709 | — | IC50 | = | 3.4 | nM | 8.47 |
| CHEMBL70 | MORPHINE | IC50 | = | - | nM | - |