Assay Detail
Binding
CHEMBL756273
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Inhibition of human ORL1 orphanin receptor
9
Total Activities
9
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
From hit to lead. Analyzing structure-profile relationships.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 9 | 6.55 | 7.72 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL115222 | — | — | 1 | 7.72 |
| CHEMBL114379 | — | — | 1 | 7.42 |
| CHEMBL115652 | — | — | 1 | 7.01 |
| CHEMBL420863 | — | — | 1 | 6.55 |
| CHEMBL326962 | — | — | 1 | 6.47 |
| CHEMBL325945 | — | — | 1 | 6.36 |
| CHEMBL325750 | — | — | 1 | 6.12 |
| CHEMBL114484 | — | — | 1 | 5.72 |
| CHEMBL115280 | — | — | 1 | 5.62 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL115222 | — | IC50 | = | 19.0 | nM | 7.72 |
| CHEMBL114379 | — | IC50 | = | 38.0 | nM | 7.42 |
| CHEMBL115652 | — | IC50 | = | 97.0 | nM | 7.01 |
| CHEMBL420863 | — | IC50 | = | 283.0 | nM | 6.55 |
| CHEMBL326962 | — | IC50 | = | 340.0 | nM | 6.47 |
| CHEMBL325945 | — | IC50 | = | 434.0 | nM | 6.36 |
| CHEMBL325750 | — | IC50 | = | 758.0 | nM | 6.12 |
| CHEMBL114484 | — | IC50 | = | 1910.0 | nM | 5.72 |
| CHEMBL115280 | — | IC50 | = | 2420.0 | nM | 5.62 |