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Assay Detail

CHEMBL756499

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibitory activity against PSPTase
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Syntheses and biological activities of a novel group of steroidal derived inhibitors for human Cdc25A protein phosphatase.
Peng H, Xie W, Otterness DM, Cogswell JP, McConnell RT, Carter HL, Powis G, Abraham RT, Zalkow LH.
J Med Chem (2001) 44 : 834 -848
PubMed 11262093 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 7.31 7.31

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL280487 OKADAIC ACID 1 7.31

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL280487 OKADAIC ACID IC50 = 49.0 nM 7.31