Assay Detail
Binding
CHEMBL758624
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Dissociation constant for binding to SH2 domain of Phosphatidylinositol 3-kinase p85 subunit
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Acquisition of high-affinity, SH2-targeted ligands via a spatially focused library.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 1 | 5.03 | 5.03 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL12253 | — | — | 1 | 5.03 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL12253 | — | Kd | = | 9300.0 | nM | 5.03 |