Assay Detail
Functional
CHEMBL759515
Review assay metadata, readout intent, target linkage, and publication context from the same page.
The compound was evaluated for antagonist activity against P2X purinoceptor 1 (P2X1) from rat vas deferens
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Purine and pyrimidine (P2) receptors as drug targets.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.07 | 5.12 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL130059 | UNIBLUE A | — | 1 | 5.12 |
| CHEMBL134193 | CIBACRON BLUE 3GA | — | 1 | 5.02 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL130059 | UNIBLUE A | IC50 | = | 7500.0 | nM | 5.12 |
| CHEMBL134193 | CIBACRON BLUE 3GA | IC50 | = | 9600.0 | nM | 5.02 |