Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL759518

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Dissociation constant of the compound at P2X purinoceptor 1 (P2X1) from rat vas deferens was reported
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

P2X purinoceptor 1 (CHEMBL2530)
Type SINGLE PROTEIN
Organism Rattus norvegicus

Publication

Purine and pyrimidine (P2) receptors as drug targets.
Jacobson KA, Jarvis MF, Williams M.
J Med Chem (2002) 45 : 4057 -4093
PubMed 12213051 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Kd 1 5.80 5.80

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL134193 CIBACRON BLUE 3GA 1 5.80

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL134193 CIBACRON BLUE 3GA Kd = 1600.0 nM 5.80