Assay Detail
Binding
CHEMBL759818
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Inhibition of enzyme pepsin
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Inhibition of aminopeptidases by peptides containing ketomethylene and hydroxyethylene amide bond replacements.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 8.00 | 8.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL28738 | — | — | 1 | 8.52 |
| CHEMBL424222 | — | — | 1 | 8.52 |
| CHEMBL28888 | — | — | 1 | 6.96 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL28738 | — | Ki | = | 3.0 | nM | 8.52 |
| CHEMBL424222 | — | Ki | = | 3.0 | nM | 8.52 |
| CHEMBL28888 | — | Ki | = | 110.0 | nM | 6.96 |