Assay Detail
Binding
CHEMBL759820
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Inhibition of pepsin
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
Designing non-peptide peptidomimetics in the 21st century: inhibitors targeting conformational ensembles.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 8.25 | 10.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3143435 | — | — | 1 | 10.00 |
| CHEMBL3143437 | — | — | 1 | 8.82 |
| CHEMBL3143436 | — | — | 1 | 5.92 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3143435 | — | Ki | = | 0.1 | nM | 10.00 |
| CHEMBL3143437 | — | Ki | = | 1.5 | nM | 8.82 |
| CHEMBL3143436 | — | Ki | = | 1200.0 | nM | 5.92 |