Assay Detail
Functional
CHEMBL762910
Review assay metadata, readout intent, target linkage, and publication context from the same page.
In vitro inhibitory activity against Prostaglandin G/H synthase 2 in IL-1-stimulated dermal fibroblasts
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
1,2-Diarylpyrroles as potent and selective inhibitors of cyclooxygenase-2.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 5.62 | 5.62 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL43664 | — | — | 1 | 5.62 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL43664 | — | IC50 | = | 2400.0 | nM | 5.62 |