Assay Detail
Functional
CHEMBL763191
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Effective concentration which increases intracellular c-AMP production in mouse EP2- receptor
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Prostaglandin E2 receptor EP2 subtype (CHEMBL2488) ↗| Type | SINGLE PROTEIN |
| Organism | Mus musculus |
Publication
Design and synthesis of a highly selective EP2-receptor agonist.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 1 | 7.48 | 7.48 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL432522 | — | — | 1 | 7.48 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL432522 | — | EC50 | = | 33.0 | nM | 7.48 |