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Assay Detail

CHEMBL763375

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Binding
Inhibitory activity against HIV-1 protease
12
Total Activities
12
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Human immunodeficiency virus 1
Confidence 9 — Direct single protein target
Curated By Expert

Target

Human immunodeficiency virus type 1 protease (CHEMBL243)
Type SINGLE PROTEIN
Organism Human immunodeficiency virus 1

Publication

Potent HIV protease inhibitors incorporating high-affinity P2-ligands and (R)-(hydroxyethylamino)sulfonamide isostere.
Ghosh AK, Kincaid JF, Cho W, Walters DE, Krishnan K, Hussain KA, Koo Y, Cho H, Rudall C, Holland L, Buthod J.
Bioorg Med Chem Lett (1998) 8 : 687 -690
PubMed 9871583 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 12 8.66 8.96

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL469086 1 8.96
CHEMBL158050 1 8.92
CHEMBL161005 1 8.92
CHEMBL161393 1 8.85
CHEMBL162086 1 8.85
CHEMBL350301 1 8.82
CHEMBL159580 1 8.82
CHEMBL116 AMPRENAVIR 4.0 1 8.80
CHEMBL1323 DARUNAVIR 4.0 1 8.68
CHEMBL422718 1 8.66
CHEMBL161644 1 8.60
CHEMBL18389 1 7.06

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL469086 Ki = 1.1 nM 8.96
CHEMBL158050 Ki = 1.2 nM 8.92
CHEMBL161005 Ki = 1.2 nM 8.92
CHEMBL161393 Ki = 1.4 nM 8.85
CHEMBL162086 Ki = 1.4 nM 8.85
CHEMBL350301 Ki = 1.5 nM 8.82
CHEMBL159580 Ki = 1.5 nM 8.82
CHEMBL116 AMPRENAVIR Ki = 1.6 nM 8.80
CHEMBL1323 DARUNAVIR Ki = 2.1 nM 8.68
CHEMBL422718 Ki = 2.2 nM 8.66
CHEMBL161644 Ki = 2.5 nM 8.60
CHEMBL18389 Ki = 87.0 nM 7.06