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Assay Detail

CHEMBL763398

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Binding
Inhibitory activity against HIV-1 protease in tandem assay.
37
Total Activities
36
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Human immunodeficiency virus 1
Confidence 9 — Direct single protein target
Curated By Expert

Target

Human immunodeficiency virus type 1 protease (CHEMBL243)
Type SINGLE PROTEIN
Organism Human immunodeficiency virus 1

Publication

Tipranavir (PNU-140690): a potent, orally bioavailable nonpeptidic HIV protease inhibitor of the 5,6-dihydro-4-hydroxy-2-pyrone sulfonamide class.
Turner SR, Strohbach JW, Tommasi RA, Aristoff PA, Johnson PD, Skulnick HI, Dolak LA, Seest EP, Tomich PK, Bohanon MJ, Horng MM, Lynn JC, Chong KT, Hinshaw RR, Watenpaugh KD, Janakiraman MN, Thaisrivongs S.
J Med Chem (1998) 41 : 3467 -3476
PubMed 9719600 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 37 9.01 10.74

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL332684 1 10.74
CHEMBL2111768 2 10.49
CHEMBL2092977 1 10.40
CHEMBL2112562 1 10.22
CHEMBL21405 1 10.00
CHEMBL2111769 1 10.00
CHEMBL2112566 1 9.92
CHEMBL2111770 1 9.92
CHEMBL116068 1 9.70
CHEMBL2111771 1 9.52
CHEMBL324579 1 9.28
CHEMBL117638 1 9.15
CHEMBL117719 1 9.06
CHEMBL116965 1 9.00
CHEMBL2092978 1 9.00
CHEMBL421230 1 8.92
CHEMBL21188 1 8.92
CHEMBL332043 1 8.77
CHEMBL118006 1 8.74
CHEMBL325454 1 8.72
CHEMBL119906 1 8.64
CHEMBL116265 1 8.59
CHEMBL117500 1 8.52
CHEMBL116798 1 8.52
CHEMBL20846 1 8.51
CHEMBL117389 1 8.37
CHEMBL326566 1 8.21
CHEMBL21281 1 8.09
CHEMBL117856 1 7.92
CHEMBL324994 1 7.89

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL332684 Ki = 0.018 nM 10.74
CHEMBL2111768 Ki = 0.032 nM 10.49
CHEMBL2092977 Ki = 0.04 nM 10.40
CHEMBL2112562 Ki = 0.06 nM 10.22
CHEMBL21405 Ki = 0.1 nM 10.00
CHEMBL2111769 Ki = 0.1 nM 10.00
CHEMBL2112566 Ki = 0.12 nM 9.92
CHEMBL2111770 Ki = 0.12 nM 9.92
CHEMBL116068 Ki = 0.2 nM 9.70
CHEMBL2111768 Ki = 0.22 nM 9.66
CHEMBL2111771 Ki = 0.3 nM 9.52
CHEMBL324579 Ki = 0.52 nM 9.28
CHEMBL117638 Ki = 0.71 nM 9.15
CHEMBL117719 Ki = 0.87 nM 9.06
CHEMBL2092978 Ki = 1.0 nM 9.00
CHEMBL116965 Ki = 1.0 nM 9.00
CHEMBL421230 Ki = 1.2 nM 8.92
CHEMBL21188 Ki = 1.2 nM 8.92
CHEMBL332043 Ki = 1.7 nM 8.77
CHEMBL118006 Ki = 1.8 nM 8.74
CHEMBL325454 Ki = 1.9 nM 8.72
CHEMBL119906 Ki = 2.3 nM 8.64
CHEMBL116265 Ki = 2.6 nM 8.59
CHEMBL117500 Ki = 3.0 nM 8.52
CHEMBL116798 Ki = 3.0 nM 8.52
CHEMBL20846 Ki = 3.1 nM 8.51
CHEMBL117389 Ki = 4.3 nM 8.37
CHEMBL326566 Ki = 6.1 nM 8.21
CHEMBL21281 Ki = 8.2 nM 8.09
CHEMBL117856 Ki = 12.0 nM 7.92
CHEMBL324994 Ki = 13.0 nM 7.89
CHEMBL115743 Ki = 17.0 nM 7.77
CHEMBL333924 Ki = 23.0 nM 7.64
CHEMBL118073 Ki = 28.0 nM 7.55
CHEMBL222559 TIPRANAVIR Ki = 0.008 nM -
CHEMBL117878 Ki > 1.0 nM -
CHEMBL2112565 Ki = 0.007 nM -