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Assay Detail

CHEMBL763761

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of phosphatidylinositol-3-kinase (P13-K)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Kinase inhibitors: not just for kinases anymore.
McGovern SL, Shoichet BK.
J Med Chem (2003) 46 : 1478 -1483
PubMed 12672248 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 8.30 8.30

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL428496 WORTMANNIN 1 8.30

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL428496 WORTMANNIN IC50 = 5.0 nM 8.30