Assay Detail

CHEMBL764561

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding

Inhibition of Phosphodiesterase 4

ChEMBL ↗

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Target

Unchecked (CHEMBL612545) ↗

Open DB target context

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Primary target Unchecked

CHEMBL612545

Anchored from Assay target.

Protein identity Unchecked

Disease frame Disease evidence pending

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Review focus Open DB context pending

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Total Activities

Compounds Tested

Activity Types

Assay Parameters

Assay Information

Assay Type	Binding
Confidence	0 — Uncurated / Unknown
Curated By	Autocuration

Target

Unchecked (CHEMBL612545) ↗

Type

UNCHECKED

Publication

Angiotensin II AT1 receptor antagonists. Clinical implications of active metabolites.

Schmidt B, Schieffer B.
J Med Chem (2003) 46 : 2261 -2270
PubMed 12773029 · DOI

Activity Statistics

Type	Count	Avg pChEMBL	Best pChEMBL
IC50	1	4.58	4.58

Compounds Tested

Compound	Name	Phase	Activities	Best pChEMBL
CHEMBL995	LOSARTAN POTASSIUM	4.0	1	4.58

Activity Data

Compound	Name	Type	Rel.	Value	Units	pChEMBL
CHEMBL995	LOSARTAN POTASSIUM	IC50	=	26000.0	nM	4.58