Assay Detail
Binding
CHEMBL765147
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of phosphorylase kinase.
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 4 — Cell-line / Tissue |
| Curated By | Expert |
Publication
Inhibitors of protein kinase C. 1. 2,3-Bisarylmaleimides.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 9.04 | 9.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL388978 | STAUROSPORINE | — | 1 | 9.30 |
| CHEMBL281948 | K-252A | — | 1 | 8.77 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL388978 | STAUROSPORINE | IC50 | = | 0.5 | nM | 9.30 |
| CHEMBL281948 | K-252A | IC50 | = | 1.7 | nM | 8.77 |