Assay Detail
Functional
CHEMBL765335
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Platelet P2T receptor antagonist activity in human platelet assay
12
Total Activities
12
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Antagonists of the platelet P2T receptor: a novel approach to antithrombotic therapy.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 12 | 8.54 | 9.48 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1160360 | — | — | 1 | 9.48 |
| CHEMBL1160361 | — | — | 1 | 9.42 |
| CHEMBL334966 | CANGRELOR | 4.0 | 1 | 9.35 |
| CHEMBL1160364 | — | — | 1 | 9.14 |
| CHEMBL1160365 | — | — | 1 | 8.87 |
| CHEMBL336292 | — | — | 1 | 8.60 |
| CHEMBL1160359 | — | — | 1 | 8.16 |
| CHEMBL1160363 | — | — | 1 | 8.02 |
| CHEMBL1160366 | — | — | 1 | 7.81 |
| CHEMBL1160357 | — | — | 1 | 6.53 |
| CHEMBL1160356 | — | — | 1 | - |
| CHEMBL1160358 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1160360 | — | IC50 | = | 0.3311 | nM | 9.48 |
| CHEMBL1160361 | — | IC50 | = | 0.3802 | nM | 9.42 |
| CHEMBL334966 | CANGRELOR | IC50 | = | 0.4467 | nM | 9.35 |
| CHEMBL1160364 | — | IC50 | = | 0.7244 | nM | 9.14 |
| CHEMBL1160365 | — | IC50 | = | 1.349 | nM | 8.87 |
| CHEMBL336292 | — | IC50 | = | 2.512 | nM | 8.60 |
| CHEMBL1160359 | — | IC50 | = | 6.918 | nM | 8.16 |
| CHEMBL1160363 | — | IC50 | = | 9.55 | nM | 8.02 |
| CHEMBL1160366 | — | IC50 | = | 15.49 | nM | 7.81 |
| CHEMBL1160357 | — | IC50 | = | 295.12 | nM | 6.53 |
| CHEMBL1160356 | — | IC50 | = | 316227.77 | nM | - |
| CHEMBL1160358 | — | IC50 | = | 316227.77 | nM | - |