Assay Detail
Binding
CHEMBL765601
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Inhibitory activity against prolyl 4-hydroxylase
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Prolyl 4-hydroxylase subunit alpha-1 (CHEMBL3301) ↗| Type | SINGLE PROTEIN |
| Organism | Rattus norvegicus |
Publication
Novel inhibitors of prolyl 4-hydroxylase. 3. Inhibition by the substrate analogue N-oxaloglycine and its derivatives.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 6.10 | 6.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL88972 | PYRIDINE-2,5-DICARBOXYLIC ACID | — | 1 | 6.10 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL88972 | PYRIDINE-2,5-DICARBOXYLIC ACID | Ki | = | 800.0 | nM | 6.10 |