Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL766046

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Parasite growth inhibition against Plasmodium falciparum FCR3
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Plasmodium falciparum
Confidence 1 — Organism
Curated By Intermediate

Target

Plasmodium falciparum (CHEMBL364)
Type ORGANISM
Organism Plasmodium falciparum

Publication

Antimalarial, antitrypanosomal, and antileishmanial activities and cytotoxicity of bis(9-amino-6-chloro-2-methoxyacridines): influence of the linker.
Girault S, Grellier P, Berecibar A, Maes L, Mouray E, Lemière P, Debreu MA, Davioud-Charvet E, Sergheraert C.
J Med Chem (2000) 43 : 2646 -2654
PubMed 10893302 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 7.72 7.77

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL330261 1 7.77
CHEMBL330260 1 7.66

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL330261 IC50 = 17.0 nM 7.77
CHEMBL330260 IC50 = 22.0 nM 7.66