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Assay Detail

CHEMBL766102

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
The compound was tested for inhibitory activity against human plasmin
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Intermediate

Target

Plasminogen (CHEMBL1801)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Discovery of LB30057, a benzamidrazone-based selective oral thrombin inhibitor.
Oh YS, Yun M, Hwang SY, Hong S, Shin Y, Lee K, Yoon KH, Yoo YJ, Kim DS, Lee SH, Lee YH, Park HD, Lee CH, Lee SK, Kim S.
Bioorg Med Chem Lett (1998) 8 : 631 -634
PubMed 9871573 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 4.32 4.32

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL7962 1 4.32

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL7962 Ki = 47900.0 nM 4.32