Assay Detail
Binding
CHEMBL766307
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Inhibition of Protein kinase C delta
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Synthesis and protein kinase C inhibitory activities of indane analogs of balanol
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 7.36 | 8.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL311399 | — | — | 1 | 8.40 |
| CHEMBL49354 | — | — | 1 | 7.30 |
| CHEMBL367488 | — | — | 1 | 6.38 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL311399 | — | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL49354 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL367488 | — | IC50 | = | 420.0 | nM | 6.38 |