Assay Detail
Binding
CHEMBL767060
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Inhibition of [3H]dofetilide binding to guinea pig cardiac potassium (K+) channels.
23
Total Activities
23
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Cavia porcellus |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Novel inhibitors of potassium ion channels on human T lymphocytes.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 23 | 6.18 | 7.24 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL53790 | — | — | 1 | 7.24 |
| CHEMBL299451 | — | — | 1 | 7.05 |
| CHEMBL416313 | — | — | 1 | 6.85 |
| CHEMBL56151 | — | — | 1 | 6.80 |
| CHEMBL56261 | — | — | 1 | 6.76 |
| CHEMBL54231 | — | — | 1 | 6.68 |
| CHEMBL59308 | — | — | 1 | 6.65 |
| CHEMBL294373 | — | — | 1 | 6.51 |
| CHEMBL293721 | — | — | 1 | 6.17 |
| CHEMBL298622 | — | — | 1 | 6.11 |
| CHEMBL53841 | — | — | 1 | 6.09 |
| CHEMBL56124 | — | — | 1 | 6.06 |
| CHEMBL56590 | — | — | 1 | 6.05 |
| CHEMBL299668 | — | — | 1 | 5.89 |
| CHEMBL291738 | — | — | 1 | 5.70 |
| CHEMBL417417 | — | — | 1 | 5.70 |
| CHEMBL298608 | — | — | 1 | 5.62 |
| CHEMBL54846 | — | — | 1 | 5.62 |
| CHEMBL54934 | — | — | 1 | 5.60 |
| CHEMBL56998 | — | — | 1 | 5.49 |
| CHEMBL56589 | — | — | 1 | 5.10 |
| CHEMBL59482 | — | — | 1 | - |
| CHEMBL53676 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL53790 | — | IC50 | = | 57.0 | nM | 7.24 |
| CHEMBL299451 | — | IC50 | = | 90.0 | nM | 7.05 |
| CHEMBL416313 | — | IC50 | = | 140.0 | nM | 6.85 |
| CHEMBL56151 | — | IC50 | = | 157.0 | nM | 6.80 |
| CHEMBL56261 | — | IC50 | = | 175.0 | nM | 6.76 |
| CHEMBL54231 | — | IC50 | = | 210.0 | nM | 6.68 |
| CHEMBL59308 | — | IC50 | = | 223.0 | nM | 6.65 |
| CHEMBL294373 | — | IC50 | = | 310.0 | nM | 6.51 |
| CHEMBL293721 | — | IC50 | = | 680.0 | nM | 6.17 |
| CHEMBL298622 | — | IC50 | = | 780.0 | nM | 6.11 |
| CHEMBL53841 | — | IC50 | = | 820.0 | nM | 6.09 |
| CHEMBL56124 | — | IC50 | = | 870.0 | nM | 6.06 |
| CHEMBL56590 | — | IC50 | = | 900.0 | nM | 6.05 |
| CHEMBL299668 | — | IC50 | = | 1300.0 | nM | 5.89 |
| CHEMBL291738 | — | IC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL417417 | — | IC50 | = | 1990.0 | nM | 5.70 |
| CHEMBL298608 | — | IC50 | = | 2400.0 | nM | 5.62 |
| CHEMBL54846 | — | IC50 | = | 2380.0 | nM | 5.62 |
| CHEMBL54934 | — | IC50 | = | 2500.0 | nM | 5.60 |
| CHEMBL56998 | — | IC50 | = | 3230.0 | nM | 5.49 |
| CHEMBL56589 | — | IC50 | = | 8000.0 | nM | 5.10 |
| CHEMBL59482 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL53676 | — | IC50 | > | 3500.0 | nM | - |