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Assay Detail

CHEMBL767430

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of Protein kinase C
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 4 — Cell-line / Tissue
Curated By Autocuration

Target

Protein kinase C (PKC) (CHEMBL2093867)
Type PROTEIN FAMILY
Organism Homo sapiens

Publication

Kinase inhibitors: not just for kinases anymore.
McGovern SL, Shoichet BK.
J Med Chem (2003) 46 : 1478 -1483
PubMed 12672248 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.61 5.61

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL16958 STAUROSPORINONE 1 5.61

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL16958 STAUROSPORINONE IC50 = 2450.0 nM 5.61