Assay Detail
Binding
CHEMBL767844
Review assay metadata, readout intent, target linkage, and publication context from the same page.
In vitro inhibitory activity against prostacyclin synthetase
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Imidazo[1,5-a]pyridines: a new class of thromboxane A2 synthetase inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 4.00 | 4.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL48092 | PIRMAGREL | 2.0 | 1 | 4.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL48092 | PIRMAGREL | IC50 | = | 100000.0 | nM | 4.00 |