Assay Detail
Functional
CHEMBL767888
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Inhibition of Platelet activating factor (PAF)- induced platelet aggregation in rabbit platelet rich plasma (PRP)
18
Total Activities
18
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Tissue | Plasma |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Novel agents combining platelet activating factor (PAF) receptor antagonist with thromboxane synthase inhibitor (TxSI).
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 18 | 7.07 | 7.50 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL349150 | — | — | 1 | 7.50 |
| CHEMBL354662 | — | — | 1 | 7.41 |
| CHEMBL165359 | — | — | 1 | 7.41 |
| CHEMBL164123 | — | — | 1 | 7.34 |
| CHEMBL350961 | — | — | 1 | 7.33 |
| CHEMBL352120 | — | — | 1 | 7.27 |
| CHEMBL323798 | — | — | 1 | 7.22 |
| CHEMBL349982 | — | — | 1 | 7.22 |
| CHEMBL351224 | — | — | 1 | 7.19 |
| CHEMBL351024 | — | — | 1 | 7.15 |
| CHEMBL164758 | — | — | 1 | 7.09 |
| CHEMBL166193 | — | — | 1 | 7.07 |
| CHEMBL351562 | — | — | 1 | 7.01 |
| CHEMBL408135 | — | — | 1 | 7.00 |
| CHEMBL166208 | — | — | 1 | 6.70 |
| CHEMBL423993 | — | — | 1 | 6.70 |
| CHEMBL424160 | — | — | 1 | 6.61 |
| CHEMBL164665 | — | — | 1 | 6.01 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL349150 | — | IC50 | = | 32.0 | nM | 7.50 |
| CHEMBL354662 | — | IC50 | = | 39.0 | nM | 7.41 |
| CHEMBL165359 | — | IC50 | = | 39.0 | nM | 7.41 |
| CHEMBL164123 | — | IC50 | = | 46.0 | nM | 7.34 |
| CHEMBL350961 | — | IC50 | = | 47.0 | nM | 7.33 |
| CHEMBL352120 | — | IC50 | = | 54.0 | nM | 7.27 |
| CHEMBL323798 | — | IC50 | = | 60.0 | nM | 7.22 |
| CHEMBL349982 | — | IC50 | = | 60.0 | nM | 7.22 |
| CHEMBL351224 | — | IC50 | = | 65.0 | nM | 7.19 |
| CHEMBL351024 | — | IC50 | = | 71.0 | nM | 7.15 |
| CHEMBL164758 | — | IC50 | = | 81.0 | nM | 7.09 |
| CHEMBL166193 | — | IC50 | = | 85.0 | nM | 7.07 |
| CHEMBL351562 | — | IC50 | = | 98.0 | nM | 7.01 |
| CHEMBL408135 | — | IC50 | = | 100.0 | nM | 7.00 |
| CHEMBL166208 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL423993 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL424160 | — | IC50 | = | 245.0 | nM | 6.61 |
| CHEMBL164665 | — | IC50 | = | 980.0 | nM | 6.01 |