Assay Detail
Binding
CHEMBL768441
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Tested for inhibition of 3[H]-iloprost binding to human IP receptor
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
A novel pyridazinone derivative as a nonprostanoid PGI2 agonist.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 7.07 | 7.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL94694 | — | — | 1 | 7.10 |
| CHEMBL94751 | — | — | 1 | 7.03 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL94694 | — | Ki | = | 80.0 | nM | 7.10 |
| CHEMBL94751 | — | Ki | = | 94.0 | nM | 7.03 |