Assay Detail
Binding
CHEMBL768532
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of protein kinase C
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 4 — Cell-line / Tissue |
| Curated By | Autocuration |
Publication
Secondary structure peptide mimetics: design, synthesis, and evaluation of beta-strand mimetic thrombin inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.69 | 5.90 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL27852 | — | — | 1 | 5.90 |
| CHEMBL282830 | — | — | 1 | 5.48 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL27852 | — | IC50 | = | 1250.0 | nM | 5.90 |
| CHEMBL282830 | — | IC50 | = | 3320.0 | nM | 5.48 |