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Assay Detail

CHEMBL769108

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Binding
Binding affinity for protein kinase C Delta-C1B domain
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Expert

Target

Protein kinase C delta type (CHEMBL2996)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Synthesis and binding selectivity of 7- and 15-decylbenzolactone-V8 for the C1 domains of protein kinase C isozymes.
Nakagawa Y, Irie K, Yamanaka N, Ohigashi H, Tsuda K.
Bioorg Med Chem Lett (2003) 13 : 3015 -3019
PubMed 12941324 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Kd 1 9.28 9.28

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL27768 1 9.28

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL27768 Kd = 0.53 nM 9.28