Assay Detail
Binding
CHEMBL769205
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Compound was evaluated for inhibitory effect against protein phosphatase I (PP-I)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Bos taurus |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Michael adducts of ascorbic acid as inhibitors of protein phosphatase 2A and inducers of apoptosis.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.24 | 5.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL40779 | — | — | 1 | 5.52 |
| CHEMBL416976 | — | — | 1 | 4.96 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL40779 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL416976 | — | IC50 | = | 11000.0 | nM | 4.96 |