Assay Detail
Functional
CHEMBL770011
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Antiproliferative activity against murine macrophage (RAW) cell line
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Cell Type | RAW |
| Confidence | 1 — Organism |
| Curated By | Expert |
Publication
Selective inhibition of the chymotrypsin-like activity of the 20S proteasome by 5-methoxy-1-indanone dipeptide benzamides.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.13 | 5.16 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL305527 | — | — | 1 | 5.16 |
| CHEMBL67885 | — | — | 1 | 5.10 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL305527 | — | IC50 | = | 7000.0 | nM | 5.16 |
| CHEMBL67885 | — | IC50 | = | 8000.0 | nM | 5.10 |