Assay Detail
Functional
CHEMBL770650
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Compound was tested for in vitro inhibition against broken RBL-1.
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Rattus norvegicus |
| Cell Type | RBL-1 |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Modulators of leukotriene biosynthesis and receptor activation.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 7.46 | 7.64 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL59356 | ATRELEUTON | 2.0 | 1 | 7.64 |
| CHEMBL90552 | — | — | 1 | 7.27 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL59356 | ATRELEUTON | IC50 | = | 23.0 | nM | 7.64 |
| CHEMBL90552 | — | IC50 | = | 54.0 | nM | 7.27 |