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Assay Detail

CHEMBL772571

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of Protein kinase C delta subunit
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Expert

Target

Protein kinase C delta type (CHEMBL2996)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Meridianins, a new family of protein kinase inhibitors isolated from the ascidian Aplidium meridianum.
Gompel M, Leost M, De Kier Joffe EB, Puricelli L, Franco LH, Palermo J, Meijer L.
Bioorg Med Chem Lett (2004) 14 : 1703 -1704
PubMed 15026054 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.92 5.92

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL296682 MERIDIANIN E 1 5.92

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL296682 MERIDIANIN E IC50 = 1200.0 nM 5.92