Assay Detail
Binding
CHEMBL798026
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Binding affinity towards human Retinoic acid receptor gamma
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Synthesis and receptor binding affinity of conformationally restricted retinoic acid analogues
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 8.36 | 9.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL38 | TRETINOIN | 4.0 | 1 | 9.22 |
| CHEMBL74331 | — | — | 1 | 7.50 |
| CHEMBL73973 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL38 | TRETINOIN | Ki | = | 0.6 | nM | 9.22 |
| CHEMBL74331 | — | Ki | = | 32.0 | nM | 7.50 |
| CHEMBL73973 | — | Ki | > | 4000.0 | nM | - |