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Assay Detail

CHEMBL798539

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antagonist binding of rN6-cyclohexyl-[3H]adenosine to rat brain
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Rattus norvegicus
Confidence 5 — Multiple protein complex / RNA
Curated By Expert

Target

Adenosine receptor (CHEMBL2111386)
Type PROTEIN FAMILY
Organism Rattus norvegicus

Publication

Adenosine receptors: targets for future drugs.
Daly JW.
J Med Chem (1982) 25 : 197 -207
PubMed 6279840 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 5.52 5.52

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL275084 ISOBUTYLMETHYLXANTHINE 1 5.52

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL275084 ISOBUTYLMETHYLXANTHINE Ki = 3000.0 nM 5.52