Assay Detail
Binding
CHEMBL799566
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Transcriptional activation of Retinoid X receptor RXR alpha;NA=not active
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Cercopithecidae |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
Synthesis and structure-activity relationships of retinoid X receptor selective diaryl sulfide analogs of retinoic acid.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 6.55 | 6.55 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL118693 | — | — | 1 | 6.55 |
| CHEMBL324960 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL118693 | — | EC50 | = | 280.0 | nM | 6.55 |
| CHEMBL324960 | — | EC50 | - | nM | - |