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Assay Detail

CHEMBL800528

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of purified recombinant human placental S-adenosyl-homocysteine hydrolase
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Adenosylhomocysteinase (CHEMBL2664)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Synthesis, mechanism of action, and antiviral activity of a new series of covalent mechanism-based inhibitors of S-adenosyl-L-homocysteine hydrolase.
Guillerm G, Guillerm D, Vandenplas-Witkowki C, Rogniaux H, Carte N, Leize E, Van Dorsselaer A, De Clercq E, Lambert C.
J Med Chem (2001) 44 : 2743 -2752
PubMed 11495586 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 3 4.65 4.80

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL607985 1 4.80
CHEMBL606446 1 4.80
CHEMBL140440 1 4.35

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL607985 Ki = 16000.0 nM 4.80
CHEMBL606446 Ki = 16000.0 nM 4.80
CHEMBL140440 Ki = 45000.0 nM 4.35