Assay Detail
Binding
CHEMBL800543
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Transcriptional activation assay in CV-1 cells expressing human retinoid X receptor RXR alpha
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | CV-1 |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Retinoic acid receptor ligands based on the 6-cyclopropyl-2,4-hexadienoic acid.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 1 | 7.89 | 7.89 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL89331 | — | — | 1 | 7.89 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL89331 | — | EC50 | = | 13.0 | nM | 7.89 |