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Assay Detail

CHEMBL800623

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibitory activity against recombinant rat liver S-adenosyl-homocysteine hydrolase
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Adenosylhomocysteinase (CHEMBL3118)
Type SINGLE PROTEIN
Organism Rattus norvegicus

Publication

Adenosine-5'-carboxaldehyde: a potent inhibitor of S-adenosyl-L-homocysteine hydrolase.
Liu S, Wnuk SF, Yuan C, Robins MJ, Borchardt RT.
J Med Chem (1993) 36 : 883 -887
PubMed 8464042 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 4 7.40 7.41

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL171700 1 7.41
CHEMBL77518 1 7.41
CHEMBL171369 1 7.40
CHEMBL308037 1 7.37

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL171700 Ki = 39.0 nM 7.41
CHEMBL77518 Ki = 39.0 nM 7.41
CHEMBL171369 Ki = 40.0 nM 7.40
CHEMBL308037 Ki = 43.0 nM 7.37