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Assay Detail

CHEMBL800723

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Exogenous inhibition concentration of Serine/threonine protein phosphatase 4 (PP4)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Serine-threonine protein phosphatase inhibitors: development of potential therapeutic strategies.
McCluskey A, Sim AT, Sakoff JA.
J Med Chem (2002) 45 : 1151 -1175
PubMed 11881984 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 9.70 9.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL280487 OKADAIC ACID 1 9.70
CHEMBL444092 MICROCYSTIN-LR 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL280487 OKADAIC ACID IC50 = 0.2 nM 9.70
CHEMBL444092 MICROCYSTIN-LR IC50 = 0.008 nM -