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Assay Detail

CHEMBL801206

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Effective concentration on human somatostatin receptor 5
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Expert

Target

Somatostatin receptor type 5 (CHEMBL1792)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Synthesis of substituted imidazopyrazines as ligands for the human somatostatin receptor subtype 5.
Contour-Galéra MO, Poitout L, Moinet C, Morgan B, Gordon T, Roubert P, Thurieau C.
Bioorg Med Chem Lett (2001) 11 : 741 -745
PubMed 11266182 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 10.19 10.19

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1823872 SOMATOSTATIN 3.0 1 10.19

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1823872 SOMATOSTATIN EC50 = 0.065 nM 10.19