Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL801228

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of [3H]ATRA binding to human Retinoic acid receptor RAR beta
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Expert

Target

Retinoic acid receptor beta (CHEMBL2008)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Retinoic acid receptor ligands based on the 6-cyclopropyl-2,4-hexadienoic acid.
Farmer LJ, Zhi L, Jeong S, Lamph WW, Osburn DL, Croston G, Flatten KS, Heyman RA, Nadzan AM.
Bioorg Med Chem Lett (2003) 13 : 261 -264
PubMed 12482435 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Kd 1 6.33 6.33

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL89331 1 6.33

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL89331 Kd = 463.0 nM 6.33