Assay Detail
Functional
CHEMBL801410
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Compound was tested for the inhibition of spermidine transporter by using [3H]SPD transport in L1210 cell
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Cell Type | L1210 |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Polyamine-iron chelator conjugate.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 4 | 5.42 | 5.77 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL82888 | — | — | 1 | 5.77 |
| CHEMBL150911 | — | — | 1 | 5.43 |
| CHEMBL284260 | — | — | 1 | 5.07 |
| CHEMBL70927 | DEFERIPRONE | 4.0 | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL82888 | — | Ki | = | 1700.0 | nM | 5.77 |
| CHEMBL150911 | — | Ki | = | 3700.0 | nM | 5.43 |
| CHEMBL284260 | — | Ki | = | 8500.0 | nM | 5.07 |
| CHEMBL70927 | DEFERIPRONE | Ki | > | 500000.0 | nM | - |